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Cayman A-61603
List Price
$36.00
Your Price
$36.00
Cayman A-61603 - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-17358-1
MFG.PART:
17358-1
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
The α1-adrenergic receptors are gq protein-coupled receptors that play a key role in the modulation of sympathetic nervous system activity and are the site of action for therapeutic agents, such as antihypertensive drugs. A-61603 is a selective α1A-adrenergic receptor agonist that is at least 35-fold more potent at α1A receptor sites than at α1B or α1D. Activation of the α1A-adrenergic receptor by A-61603 has been reported to increase the frequency of spontaneous Ca2+ transients in rat ventricular myocytes in vitro (EC50 = 6.9 nM) much more potently than activation by phenylephrine (Item No. ; EC50 = 2.3 µM).
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
N-[5-(4,5-dihydro-1H-imidazol-2-yl)-5,6,7,8-tetrahydro-2-hydroxy-1-naphthalenyl]-methanesulfonamide, monohydrobromide
CAS Number
107756-30-9
Molecular Formula
C14H19N3O3S • HBr
Formula Weight
390.3
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 20 mg/mL
- DMSO: 20 mg/mL
- Ethanol: 1 mg/mL
- PBS (pH 7.2): 10 mg/mL
SMILES
OC1=C(NS(C)(=O)=O)C2=C(C(C3=NCCN3)CCC2)C=C1.Br
InChi Code
InChI=1S/C14H19N3O3S.BrH/c1-21(19,20)17-13-10-3-2-4-11(14-15-7-8-16-14)9(10)5-6-12(13)18;/h5-6,11,17-18H,2-4,7-8H2,1H3,(H,15,16);1H
InChi Key
LRFLWCZMTGTUEP-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-17358-1 |
|---|---|
| Supplier Part Number | 17358-1 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer Name | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 107756-30-9 |
| Energy Star | No |
| Green | No |
| Controlled | N |