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Cayman Tcs-Ox2-29; Purity- Greater Than Or Equal To 98%; Size- 50
List Price
$768.00
Your Price
$768.00
Cayman Tcs-Ox2-29; Purity- Greater Than Or Equal To 98%; Size- 50 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-17419-50
MFG.PART:
17419-50
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
Orexin receptors R1 (OX1R) and OX2R mediate the action of the neuropeptides orexin A and orexin B. TCX-OX2-29 is an antagonist of OX2R (pKi = 7.5) that exhibits >250-fold selectivity for hOX2R compared with hOX1R (IC50s = 40 nM and >10,000 nM, respectively).1,2 It blocks the inhibitory action of orexin A on forskolin-induced cAMP formation.3
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
(2S)-1-(3,4-dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)-3,3-dimethyl-2-[(4-pyridinylmethyl)amino]-1-butanone, monohydrochloride
CAS Number
1610882-30-8
Molecular Formula
C23H31N3O3 • HCl
Formula Weight
434.0
Purity
≥95%
Formulation(Request formulation change)
A crystalline solid
Solubility(Learn about Variance in Solubility)
- DMF: 30 mg/ml
- DMSO: 30 mg/ml
- PBS (pH 7.2): 10 mg/ml
λmax
286 nm
SMILES
COC1=C(OC)C=C(CN(C([C@H](C(C)(C)C)NCC2=CC=NC=C2)=O)CC3)C3=C1.Cl
InChi Code
InChI=1S/C23H31N3O3.ClH/c1-23(2,3)21(25-14-16-6-9-24-10-7-16)22(27)26-11-8-17-12-19(28-4)20(29-5)13-18(17)15-26;/h6-7,9-10,12-13,21,25H,8,11,14-15H2,1-5H3;1H/t21-;/m1./s1
InChi Key
NHKNHFJTMINMBP-ZMBIFBSDSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Wet ice in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-17419-50 |
|---|---|
| Featured | No |
| Supplier Part Number | 17419-50 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Refrigerated |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 2 |
| Hazardous | N |
| CAS Number | 1610882-30-8 |
| Energy Star | No |
| Green | No |
| ACT Ecolabel | No |
| Controlled | N |