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Cayman Gs967; Purity- Greater Than Or Equal To 98%; Size- 50 Mg;
List Price
$146.00
Your Price
$146.00
Cayman Gs967; Purity- Greater Than Or Equal To 98%; Size- 50 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-18376-50
MFG.PART:
18376-50
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
Inhibition of cardiac late sodium current (late INa) is a strategy to suppress arrhythmias and sodium-dependent calcium overload associated with myocardial ischemia and heart failure. GS967 is a selective inhibitor of late INa that has been shown to suppress experimentally induced arrhythmias in rabbit myocytes and hearts.1 It can inhibit A. sulcata toxin II–induced late INa in ventricular myocytes and isolated hearts with IC50 values of 0.13 and 0.21 µM, respectively.1 GS967 causes minimal inhibition of the delayed-rectifier potassium current nor does it affect L- or T-type calcium channel currents, sodium-calcium exchanger currents, or a panel of 162 receptors, ion channels, transporters, and enzymes.1
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
6-[4-
CAS Number
1262618-39-2
Molecular Formula
C14H7F6N3O
Formula Weight
347.2
Purity
≥98%
Formulation(Request formulation change)
A crystalline solid
Solubility(Learn about Variance in Solubility)
- DMF: 25 mg/ml
- DMF:PBS(pH7.2) (1:2): 0.3 mg/ml
- DMSO: 20 mg/ml
- Ethanol: 12 mg/ml
λmax
247 nm
SMILES
FC(OC1=CC=C(C(C=C2)=CN3C2=NN=C3C(F)(F)F)C=C1)(F)F
InChi Code
InChI=1S/C14H7F6N3O/c15-13(16,17)12-22-21-11-6-3-9(7-23(11)12)8-1-4-10(5-2-8)24-14(18,19)20/h1-7H
InChi Key
FEVBKJITJDHASC-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-18376-50 |
|---|---|
| Featured | No |
| Supplier Part Number | 18376-50 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Refrigerated |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 2 |
| Hazardous | N |
| CAS Number | 1262618-39-2 |
| Energy Star | No |
| Green | No |
| ACT Ecolabel | No |
| Controlled | N |