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Cayman (±)-WIN 55,212 (mesylate)
List Price $124.00 Your Price $124.00
Cayman (±)-WIN 55,212 (mesylate) - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-10736-10
MFG.PART: 10736-10
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
(±)-WIN 55,212 is a racemic mixture of the cannabinoid (CB) receptor 1 (CB1) and CB2 agonist (+)-WIN 55,212-2 (Item No. ) and the CB2 neutral antagonist (−)-WIN 55,212-3 (Item No. ). It inhibits electrically induced contractions in mouse vas deferens preparations (IC50 = 0.006 µM) and reduces prostaglandin (PG) synthesis by 35% in mouse brain microsomes when used at a concentration of 30 µM. (±)-WIN 55,212 decreases acetylcholine-induced writhing in mice with an ED50 value of 0.25 mg/kg. It induces hypolocomotion, analgesia, hypothermia, and catalepsy in mice (ED50s = 1.09, 0.5, 3.01 and 6.8 mg/kg, respectively).
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
[2,3-
CAS Number
137795-17-6
Molecular Formula
C27H26N2O3 • CH3SO3H
Formula Weight
522.6
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 30 mg/mL
- DMSO: 30 mg/mL
- DMSO:PBS (pH 7.2) (1:2): 0.25 mg/mL
- Ethanol: 5 mg/mL
- Methanol: 1 mg/mL
λmax
220, 331 nm
SMILES
O=C(C1=CC=CC2=C1C=CC=C2)C3=C(C)N(C4=C3C=CC=C4OC5)C5CN6CCOCC6.CS(=O)(O)=O
InChi Code
InChI=1S/C27H26N2O3.CH4O3S/c1-18-25(27(30)22-9-4-7-19-6-2-3-8-21(19)22)23-10-5-11-24-26(23)29(18)20(17-32-24)16-28-12-14-31-15-13-28;1-5(2,3)4/h2-11,20H,12-17H2,1H3;1H3,(H,2,3,4)
InChi Key
FSGCSTPOPBJYSX-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-10736-10 |
|---|---|
| Supplier Part Number | 10736-10 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 137795-17-6 |
| Energy Star | No |
| Green | No |
| Controlled | N |