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Cayman SER-601
List Price $194.00 Your Price $194.00
Cayman SER-601 - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-11743-10
MFG.PART: 11743-10
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
SER-601 is a potent and selective peripheral cannabinoid (CB2) receptor agonist with 190-fold selectivity for CB2 over the central CB1 receptor (Kis = 6.3 and 1,220 nM, respectively)., At 3 mg/kg, SER-601 has analgesic effects in a formalin-induced nocifensive study in mice without cannabis-like behavioral effects due to its low affinity for the CB1 receptor., SER-601 also has antidiabetic effects. Two to four week exposure to SER-601 ameliorates insulin resistance in vivo and increases insulin secretion and accumulation in pancreatic islets isolated from high-fat diet/streptozotocin (HFD/STZ)-induced diabetic mice.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
1,4-
CAS Number
1048038-90-9
Molecular Formula
C28H38N2O2
Formula Weight
434.6
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 5 mg/mL
- Ethanol: 3 mg/mL
λmax
217, 250, 258, 307, 323, 335 nm
SMILES
CC(C)C1=CC2=C(N(CCCCC)C=C(C(NC3(C[C@H]4C5)C[C@@H](C4)C[C@@H]5C3)=O)C2=O)C=C1
InChi Code
InChI=1S/C28H38N2O2/c1-4-5-6-9-30-17-24(26(31)23-13-22(18(2)3)7-8-25(23)30)27(32)29-28-14-19-10-20(15-28)12-21(11-19)16-28/h7-8,13,17-21H,4-6,9-12,14-16H2,1-3H3,(H,29,32)/t19-,20+,21-,28?
InChi Key
KUMKLUDNETVLDS-XMURTRJZSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-11743-10 |
|---|---|
| Supplier Part Number | 11743-10 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 1048038-90-9 |
| Energy Star | No |
| Green | No |
| Controlled | N |