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Cayman RP-8-CPT-Cyclic AMP (sodium salt)
List Price $380.00 Your Price $380.00
Cayman RP-8-CPT-Cyclic AMP (sodium salt) - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-17142-1
MFG.PART: 17142-1
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
RP-8-CPT-cAMP is a structural combination of the lipophilic and non-hydrolyzable cAMP analogs, 8-CPT-cyclic AMP (Item No. ) and RP-cyclic AMPS (Item No. ). It functions as a site-selective inhibitor of protein kinase A (PKA) type I and II, with preference towards site A of type I and site B of type II. By occupying cAMP binding sites at the regulatory subunit of PKA, RP-8-CPT-cAMP prevents the kinase holoenzyme from dissociative activation.,
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
8-[(4-
CAS Number
221905-35-7
Synonyms
- RP-8-CPT
-cAMP
Molecular Formula
C16H14ClN5O5PS2 • Na
Formula Weight
509.8
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 30 mg/mL
- DMSO: 25 mg/mL
- Ethanol: 0.5 mg/mL
- PBS (pH 7.2): 10 mg/mL
λmax
275 nm
SMILES
O[C@H]1[C@H](N2C(SC3=CC=C(Cl)C=C3)=NC4=C2N=CN=C4N)O[C@H]5[C@H]1O[P@@](OC5)([S-])=O.[Na+]
InChi Code
InChI=1S/C16H15ClN5O5PS2.Na/c17-7-1-3-8(4-2-7)30-16-21-10-13(18)19-6-20-14(10)22(16)15-11(23)12-9(26-15)5-25-28(24,29)27-12;/h1-4,6,9,11-12,15,23H,5H2,(H,24,29)(H2,18,19,20);/q;+1/p-1/t9-,11-,12-,15-,28-;/m1./s1
InChi Key
AWXMSJRRXLCVMW-ALHPSJIMSA-M
Shipping & Storage Information
Storage
-20°C
Shipping
Wet ice in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-17142-1 |
|---|---|
| Supplier Part Number | 17142-1 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | Germany |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 221905-35-7 |
| Energy Star | No |
| Green | No |
| Controlled | N |