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Cayman DA-3003-2
List Price $69.00 Your Price $69.00
Cayman DA-3003-2 - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-17282-1
MFG.PART: 17282-1
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
Cdc25 dual-specific protein tyrosine phosphatases are important for cell cycle progression and often overexpressed in cancers. Through the removal of inhibitory phosphates, they function to catalyze the activation of cyclin-Cdk complexes. DA-3003-2 is a Cdc25 phosphatase inhibitor (IC50 = 0.82 µM for human recombinant Cdc25B) that demonstrates antiproliferative activity.,, At 20 µM, it has been shown to arrest asynchronous PC-3 prostate cancer cells in g2/M phase.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
7-chloro-6-
CAS Number
383907-47-9
Synonyms
- NSC 663285
Molecular Formula
C15H16ClN3O3
Formula Weight
321.8
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 30 mg/mL
- DMSO: 20 mg/mL
λmax
233, 272, 477 nm
SMILES
O=C(C(NCCN1CCOCC1)=C2Cl)C3=C(N=CC=C3)C2=O
InChi Code
InChI=1S/C15H16ClN3O3/c16-11-13(18-4-5-19-6-8-22-9-7-19)14(20)10-2-1-3-17-12(10)15(11)21/h1-3,18H,4-9H2
InChi Key
LGTBDMBBPVNDSZ-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-17282-1 |
|---|---|
| Supplier Part Number | 17282-1 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 383907-47-9 |
| Energy Star | No |
| Green | No |
| Controlled | N |