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Cayman Solifenacin (Succinate); Purity- Greater Than Or Equal To
List Price
$48.00
Your Price
$48.00
Cayman Solifenacin (Succinate); Purity- Greater Than Or Equal To 98%; Size- 25 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-17320-25
MFG.PART:
17320-25
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
Solifenacin is a competitive antagonist of M1, M2, and M3 muscarinic acetylcholine receptors (Kis = 25, 125, and 10 nM, respectively, for the human receptors).1 It inhibits calcium mobilization induced by carbachol (carbamoylcholine; Item No. 14486) in isolated guinea pig detrusor muscle cells (Ki = 4 nM).2 Solifenacin inhibits carbachol-induced contraction of isolated guinea pig urinary bladder smooth muscle. In vivo, solifenacin (0.03-1 mg/kg) inhibits carbachol-induced increases in urinary bladder pressure in anesthetized rats. Formulations containing solifenacin have been used in the treatment of overactive bladder.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
butanedioic acid, compd. with (1S)-(3R)-1- azabicyclo [2.2.2]oct-3- yl 3,4-di hydro-1- phenyl-2(1H)- isoquinoline carboxylate
CAS Number
242478-38-2
Synonyms
- YM-67905
Molecular Formula
C23H26N2O2 • C4H6O4
Formula Weight
480.6
Purity
≥98%
Formulation(Request formulation change)
A crystalline solid
Solubility(Learn about Variance in Solubility)
- DMF: 25 mg/ml
- DMSO: 25 mg/ml
- Ethanol: 5 mg/ml
- PBS (pH 7.2): 10 mg/ml
SMILES
O=C(O[C@H]1CN2CCC1CC2)N3[C@@H](C4=CC=CC=C4)C5=CC=CC=C5CC3.OC(CCC(O)=O)=O
InChi Code
InChI=1S/C23H26N2O2.C4H6O4/c26-23(27-21-16-24-13-10-18(21)11-14-24)25-15-12-17-6-4-5-9-20(17)22(25)19-7-2-1-3-8-19;5-3(6)1-2-4(7)8/h1-9,18,21-22H,10-16H2;1-2H2,(H,5,6)(H,7,8)/t21-,22-;/m0./s1
InChi Key
RXZMMZZRUPYENV-VROPFNGYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-17320-25 |
|---|---|
| Featured | No |
| Supplier Part Number | 17320-25 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Refrigerated |
| CountryOfOrigin | China |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 2 |
| Hazardous | N |
| CAS Number | 242478-38-2 |
| Energy Star | No |
| Green | No |
| ACT Ecolabel | No |
| Controlled | N |