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Cayman Cox-1 (Human Recombinant); Purity- Greater Than Or Equal T
List Price
$820.00
Your Price
$820.00
Cayman Cox-1 (Human Recombinant); Purity- Greater Than Or Equal To 85% Estimated By Sds-Page; Size- 5 Kunits; - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-17616-5
MFG.PART:
17616-5
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
SB 277011A is an antagonist of the dopamine D3 receptor (pKi = 8.0) that is at least 100-fold selective for D3 over other monoamine receptors (pKis = 6.0, 5.0, and <5.2 for D2, 5-HT1D and 5-HT1B respectively).,, It has high oral bioavailability and enters the central nervous system of the rat. SB 277011A has been shown to have potential benefits in animal models of schizophrenia and Parkinson’s disease.,
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
N- [trans- 4- [2- (6- cyano- 3,4- di hydro- 2(1H)- iso quinolinyl) ethyl] cyclo hexyl]- 4- quinoline carbox amide, dihydro chloride
CAS Number
1226917-67-4
Molecular Formula
C28H30N4O • 2HCl
Formula Weight
511.5
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 3 mg/ml
- DMSO: 14 mg/ml
- DMSO:PBS (pH 7.2)(1:9): 0.1 mg/ml
- Ethanol: 0.1 mg/ml
λmax
230, 284 nm
SMILES
O=C(C1=C2C(C=CC=C2)=NC=C1)N[C@H](CC3)CC[C@@H]3CCN(C4)CCC5=C4C=CC(C#N)=C5.Cl.Cl
InChi Code
InChI=1S/C28H30N4O.2ClH/c29-18-21-5-8-23-19-32(16-13-22(23)17-21)15-12-20-6-9-24(10-7-20)31-28(33)26-11-14-30-27-4-2-1-3-25(26)27;;/h1-5,8,11,14,17,20,24H,6-7,9-10,12-13,15-16,19H2,(H,31,33);2*1H/t20-,24-;;
InChi Key
HEZIOTGUXSPDAK-ONAIBGCWSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-17616-5 |
|---|---|
| Featured | No |
| Supplier Part Number | 17616-5 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -80 |
| Refrigerated-Frozen | Frozen |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 2 |
| Hazardous | N |
| Energy Star | No |
| Green | No |
| ACT Ecolabel | No |
| Controlled | N |