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Cayman Ml-299; Purity- Greater Than Or Equal To 95%; Size- 5 Mg;
List Price
$437.00
Your Price
$437.00
Cayman Ml-299; Purity- Greater Than Or Equal To 95%; Size- 5 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-17632-5
MFG.PART:
17632-5
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
ML-299 is a dual inhibitor of phospholipase D1 (PLD1) and PLD2 (IC50s = 6 and 20 nM, respectively).1 It is selective for PLD1 and PLD2 over a panel of 65 receptors but also inhibits human-ether-a-go-go (hERG), also known as Kv11.1, as well as κ- and µ-opioid receptors at 10 µM.2 ML-299 (1 and 10 µM) decreases invasive migration of U87MG glioblastoma cells.1
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
4-bromo-N- [(1S)-2-[1-(3- fluorophenyl)- 4-oxo-1,3,8- triazaspiro [4.5]dec-8- yl]-1- methylethyl]- benzamide
CAS Number
1426916-00-8
Synonyms
- CID-56593087
Molecular Formula
C23H26BrFN4O2
Formula Weight
489.4
Purity
≥95%
Formulation(Request formulation change)
A crystalline solid
Solubility(Learn about Variance in Solubility)
- DMF: 30 mg/ml
- DMF:PBS (pH 7.2) (1:20): 0.5 mg/ml
- DMSO: 25 mg/ml
- Ethanol: 1 mg/ml
λmax
247 nm
SMILES
BrC1=CC=C(C(N[C@@H](C)CN2CCC3(C(NCN3C4=CC(F)=CC=C4)=O)CC2)=O)C=C1
InChi Code
InChI=1S/C23H26BrFN4O2/c1-16(27-21(30)17-5-7-18(24)8-6-17)14-28-11-9-23(10-12-28)22(31)26-15-29(23)20-4-2-3-19(25)13-20/h2-8,13,16H,9-12,14-15H2,1H3,(H,26,31)(H,27,30)/t16-/m0/s1
InChi Key
RFKXAYJUFUZBMA-INIZCTEOSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-17632-5 |
|---|---|
| Featured | No |
| Supplier Part Number | 17632-5 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Refrigerated |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 2 |
| Hazardous | N |
| CAS Number | 1426916-00-8 |
| Energy Star | No |
| Green | No |
| ACT Ecolabel | No |
| Controlled | N |