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Cayman Tasquinimod; Purity- Greater Than Or Equal To 98%; Size- 5
List Price
$202.00
Your Price
$202.00
Cayman Tasquinimod; Purity- Greater Than Or Equal To 98%; Size- 5 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-17692-5
MFG.PART:
17692-5
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
TG11-77 is a brain-permeable antagonist of the prostaglandin E2 (PGE2) receptor subtype EP2 (KB = 9.7 nM). It is selective for EP2 over DP1, EP4, and IP receptors (KBs = 7,320, 5,300, and >10,000 nM, respectively). TG11-77 (0.3 and 1 μM) inhibits the expression of genes encoding COX-2, IL-1β, and IL-6 induced by LPS and the EP2 receptor agonist ONO-AE1-259-01 in mouse BV-2 microglia expressing human EP2 receptors.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
2-((4,6- dimethyl pyridin-2-yl) amino)-N-(2- (2-methyl-1H- indol-3-yl) ethyl) pyrimidine-5- carboxamide, monohydro chloride
CAS Number
2550393-38-7
Molecular Formula
C23H24N6O • HCl
Formula Weight
436.9
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMSO: 10 mg/ml
- DMSO:PBS (pH 7.2) (1:2): 0.33 mg/ml
λmax
225, 261, 324 nm
SMILES
O=C(C1=CN=C(NC2=NC(C)=CC(C)=C2)N=C1)NCCC3=C(C)NC4=C3C=CC=C4.Cl
InChi Code
InChI=1S/C23H24N6O.ClH/c1-14-10-15(2)27-21(11-14)29-23-25-12-17(13-26-23)22(30)24-9-8-18-16(3)28-20-7-5-4-6-19(18)20;/h4-7,10-13,28H,8-9H2,1-3H3,(H,24,30)(H,25,26,27,29);1H
InChi Key
KNHQNXHZXZHWSS-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Wet ice in continental US; may vary elsewhere
Stability
≥ 2 years
| SKU | CAYM-17692-5 |
|---|---|
| Featured | No |
| Supplier Part Number | 17692-5 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Refrigerated |
| CountryOfOrigin | China |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 2 |
| Hazardous | N |
| CAS Number | 254964-60-8 |
| Energy Star | No |
| Green | No |
| ACT Ecolabel | No |
| Controlled | N |