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Cayman SR 49059
List Price $54.00 Your Price $54.00
Cayman SR 49059 - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-17972-1
MFG.PART: 17972-1
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
SR 49059 is a selective, nonpeptide antagonist of the V1a subtype of the vasopressin receptor (Ki = 1.1-6.3 nM in human)., It demonstrates ≥2 orders of magnitude lower affinity for V1b, V2, and oxytocin receptors and does not exhibit any intrinsic agonist activity. SR 49059 can inhibit arginine vasopressin-induced human platelet aggregation with an IC50 value of 3.7 nM.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
1-[[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-2-pyrrolidinecarboxamide
CAS Number
150375-75-0
Synonyms
- Relcovaptan
Molecular Formula
C28H27Cl2N3O7S
Formula Weight
620.5
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 5 mg/mL
- DMSO: 5 mg/mL
- Ethanol: 5 mg/mL
SMILES
ClC1=CC=CC=C1[C@]2(O)[C@H](C(N3CCC[C@H]3C(N)=O)=O)N(S(C4=CC=C(OC)C(OC)=C4)(=O)=O)C5=CC=C(Cl)C=C52
InChi Code
InChI=1S/C28H27Cl2N3O7S/c1-39-23-12-10-17(15-24(23)40-2)41(37,38)33-21-11-9-16(29)14-19(21)28(36,18-6-3-4-7-20(18)30)25(33)27(35)32-13-5-8-22(32)26(31)34/h3-4,6-7,9-12,14-15,22,25,36H,5,8,13H2,1-2H3,(H2,31,34)/t22-,25-,28+/m0/s1
InChi Key
CEBYCSRFKCEUSW-NAYZPBBASA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-17972-1 |
|---|---|
| Supplier Part Number | 17972-1 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | Canada |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 150375-75-0 |
| Energy Star | No |
| Green | No |
| Controlled | N |