We use cookies to make your experience better. To comply with the new e-Privacy directive, we need to ask for your consent to set the cookies. Learn more.
Cayman Adp-Glucose (Sodium Salt); Purity- Greater Than Or Equal T
List Price
$47.00
Your Price
$47.00
Cayman Adp-Glucose (Sodium Salt); Purity- Greater Than Or Equal To 95%; Size- 5 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-18139-5
MFG.PART:
18139-5
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
The indole derivative SB-207266 is a selective and potent antagonist of the serotonin (5-HT) receptor 5-HT4 with a pA2 value of 10.6 ± 0.1., In COS7 cells, 100 nM SB-207266 inhibited 5-HT4 responses to 5-HT and reduced basal agonist-independent cAMP production. In several animal models, low concentrations of SB-207266 blocked exogenous 5-HT-mediated sensitization of intestinal peristalsis.,, In a dog model, SB-207266 (0.1–100 pg/kg) dose-dependently reduced responses to 5-HT, with an ID50 value of 1.3 pg/kg. SB-206226 (0.5 mg/kg/24 h) improved cardiac function in a rat model of congestive heart failure.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
N-[(1-butyl- 4-piperidinyl )methyl]-3,4- dihydro-2H- [1,3]oxazino [3,2-a]indole -10- carboxamide
CAS Number
152811-62-6
Synonyms
- Piboserod
Molecular Formula
C22H31N3O2
Formula Weight
369.5
Purity
≥95%
Formulation
A crystalline solid
Solubility
- DMF: 30 mg/mL
- DMSO: 20 mg/mL
- Ethanol: 30 mg/mL
- Ethanol:PBS (pH7.2)(1:20): 0.05 mg/mL
λmax
224, 263, 294 nm
SMILES
CCCCN1CCC(CNC(C2=C3N(CCCO3)C4=C2C=CC=C4)=O)CC1
InChi Code
InChI=1S/C22H31N3O2/c1-2-3-11-24-13-9-17(10-14-24)16-23-21(26)20-18-7-4-5-8-19(18)25-12-6-15-27-22(20)25/h4-5,7-8,17H,2-3,6,9-16H2,1H3,(H,23,26)
InChi Key
KVCSJPATKXABRQ-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-18139-5 |
|---|---|
| Featured | No |
| Supplier Part Number | 18139-5 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Refrigerated |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 2 |
| Hazardous | N |
| CAS Number | 102129-65-7 |
| Energy Star | No |
| Green | No |
| ACT Ecolabel | No |
| Controlled | N |