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Cayman NVS-CECR2-1
List Price $90.00 Your Price $90.00
Cayman NVS-CECR2-1 - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-18316-1
MFG.PART: 18316-1
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
NVS-CECR2-1 is a potent inhibitor of CECR2 (cat eye syndrome chromosome region, candidate 2), a component of chromatin complexes that regulate gene expression controlling development. It binds CECR2 with high affinity (IC50 = 0.047 µM by Alpha screen, Kd = 0.80 µM by ITC). NVS-CECR2-1 demonstrates no crossreactivity in a panel of 48 bromodomains and has no major activity in kinase, protease, and receptor panels. It shows robust activity in cells by FRAP assay, due to its slow off-rate, and has no acute toxicity. See the website for more information.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
N-cyclopropyl-
CAS Number
1992047-61-6
Synonyms
- NVS-1
Molecular Formula
C27H37N5O2S
Formula Weight
495.7
Purity
≥95%
Formulation
A crystalline solid
Solubility
- DMSO: 0.3 mg/mL
λmax
267 nm
SMILES
O=S(C1=NC(NC2CC2)=CC(C3=CC(C=CN4C5CC(C)(C)NC(C)(C)C5)=C4C=C3)=N1)(CCC)=O
InChi Code
InChI=1S/C27H37N5O2S/c1-6-13-35(33,34)25-29-22(15-24(30-25)28-20-8-9-20)18-7-10-23-19(14-18)11-12-32(23)21-16-26(2,3)31-27(4,5)17-21/h7,10-12,14-15,20-21,31H,6,8-9,13,16-17H2,1-5H3,(H,28,29,30)
InChi Key
XVECNLUKQDKOST-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-18316-1 |
|---|---|
| Supplier Part Number | 18316-1 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 1992047-61-6 |
| Energy Star | No |
| Green | No |
| Controlled | N |