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Cayman Wye-125132; Purity- Greater Than Or Equal To 98%; Size- 10
List Price
$186.90
Your Price
$186.90
Cayman Wye-125132; Purity- Greater Than Or Equal To 98%; Size- 10 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-18372-10
MFG.PART:
18372-10
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
GSK4027 is a p300/CBP-associated factor (PCAF)/general control nonderepressible 5 (GCN5) bromodomain inhibitor (Ki = 1.4 nM; IC50 = 60 nM in a chromatin engagement assay). It is greater than 18,000-fold selective for PCAF and GCN5 over BET family bromodomains and greater than 70-fold selective over other bromodomain families in a BROMOscan assay.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
4-bromo-2-
CAS Number
2079896-25-4
Molecular Formula
C17H21BrN4O
Formula Weight
377.3
Purity
≥95%
Formulation
A crystalline solid
Solubility
- DMSO: soluble
λmax
228, 292 nm
SMILES
CN1C[C@@H](C2=CC=CC=C2)C[C@@H](NC(C=NN3C)=C(Br)C3=O)C1
InChi Code
InChI=1S/C17H21BrN4O/c1-21-10-13(12-6-4-3-5-7-12)8-14(11-21)20-15-9-19-22(2)17(23)16(15)18/h3-7,9,13-14,20H,8,10-11H2,1-2H3/t13-,14+/m0/s1
InChi Key
VZAFGXCWAWRULT-UONOGXRCSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-18372-10 |
|---|---|
| Featured | No |
| Supplier Part Number | 18372-10 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Refrigerated |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 2 |
| Hazardous | N |
| CAS Number | 1144068-46-1 |
| Energy Star | No |
| Green | No |
| ACT Ecolabel | No |
| Controlled | N |