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Cayman DREADD Agonist 21
List Price $53.00 Your Price $53.00
Cayman DREADD Agonist 21 - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-18907-1
MFG.PART: 18907-1
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
DREADD agonist 21 activates hM3Dq (EC50 = 1.7 nM), a designer receptor exclusively activated by designer drugs (DREADD) derived from the human muscarinic acetylcholine M3 receptor. It does not agonize the hM3 receptor and displays relatively weaker binding affinities for serotonin 5-HT2A, 5-HT2C, α1A-adrenergic, and histamine H1 receptors (Kis = 66, 170, 280, and 6 nM, respectively).
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
11-(1-
CAS Number
56296-18-5
Molecular Formula
C17H18N4
Formula Weight
278.4
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 10 mg/mL
- DMSO: 10 mg/mL
- DMSO:PBS(pH7.2) (1:1): 0.5 mg/mL
- Ethanol: 5 mg/mL
λmax
224, 295 nm
SMILES
C1(C=CC=C2)=C2NC(C=CC=C3)=C3C(N4CCNCC4)=N1
InChi Code
InChI=1S/C17H18N4/c1-2-6-14-13(5-1)17(21-11-9-18-10-12-21)20-16-8-4-3-7-15(16)19-14/h1-8,18-19H,9-12H2
InChi Key
JCBYXNSOLUVGTF-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-18907-1 |
|---|---|
| Supplier Part Number | 18907-1 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 56296-18-5 |
| Energy Star | No |
| Green | No |
| Controlled | N |