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Cayman Prt4165; Purity- Greater Than Or Equal To 98%; Size- 5 Mg
List Price
$57.00
Your Price
$57.00
Cayman Prt4165; Purity- Greater Than Or Equal To 98%; Size- 5 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-19093-5
MFG.PART:
19093-5
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
Exchange protein activated by cAMP (Epac) proteins mediate cAMP signaling independent of protein kinase A (PKA). ESI-09 is an inhibitor of Epac1 and Epac2 with IC50 values of 3.2 and 1.4 µM, respectively. It shows no activity against PKA at concentrations as high as 25 µM., ESI-09 has been shown to block Akt phosphorylation and insulin secretion in pancreatic β cells, as well as to block the migration of AsPC-1 and PANC-1 pancreatic cancer cells in vitro.,
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
α-[2-(3-chlorophenyl)
CAS Number
263707-16-0
Molecular Formula
C16H15ClN4O2
Formula Weight
330.8
Purity
≥95%
Formulation
A crystalline solid
Solubility
- DMF: 5 mg/ml
- DMSO: 10 mg/ml
- DMSO:PBS (pH 7.2) (1:7): 0.1 mg/ml
- Ethanol: 1 mg/ml
λmax
252, 367 nm
SMILES
ClC1=CC=CC(N/N=C(C#N)/C(C2=NOC(C(C)(C)C)=C2)=O)=C1
InChi Code
InChI=1S/C16H15ClN4O2/c1-16(2,3)14-8-12(21-23-14)15(22)13(9-18)20-19-11-6-4-5-10(17)7-11/h4-8,19H,1-3H3/b20-13+
InChi Key
DXEATJQGQHDURZ-DEDYPNTBSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-19093-5 |
|---|---|
| Featured | No |
| Supplier Part Number | 19093-5 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Refrigerated |
| CountryOfOrigin | China |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 2 |
| Hazardous | N |
| CAS Number | 31083-55-3 |
| Energy Star | No |
| Green | No |
| ACT Ecolabel | No |
| Controlled | N |