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Cayman TP-064
List Price
$36.00
Your Price
$36.00
Cayman TP-064 - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-20256-1
MFG.PART:
20256-1
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
TP-064 is a potent inhibitor of protein arginine methyltransferase 4 (PRMT4; IC50 < 10 nM) that is greater than 100-fold selective over other histone methyltransferases and non-epigenetic targets. It also inhibits methylation of the RNA polymerase II mediator complex subunit 12 (MED12; IC50 = 43 nM) in vitro. For more information on TP-064 please visit the . The negative control, TP-064N, for TP-064 is also available exclusively through the SGC. You can submit a request to receive the negative control .
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
N-methyl-N- [[2-[1-[2- (methylamino) ethyl]-4- piperidinyl]- 4-pyridinyl] methyl]-3- phenoxy- benzamide
CAS Number
2080306-20-1
Molecular Formula
C28H34N4O2
Formula Weight
458.6
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 30 mg/mL
- DMSO: 30 mg/mL
- Ethanol: 30 mg/mL
SMILES
O=C(N(CC1=CC(C2CCN(CCNC)CC2)=NC=C1)C)C3=CC=CC(OC4=CC=CC=C4)=C3
InChi Code
InChI=1S/C28H34N4O2/c1-29-15-18-32-16-12-23(13-17-32)27-19-22(11-14-30-27)21-31(2)28(33)24-7-6-10-26(20-24)34-25-8-4-3-5-9-25/h3-11,14,19-20,23,29H,12-13,15-18,21H2,1-2H3
InChi Key
VUIITYLFSAXKIQ-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-20256-1 |
|---|---|
| Supplier Part Number | 20256-1 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 2080306-20-1 |
| Energy Star | No |
| Green | No |
| Controlled | N |