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Cayman Vilanterol
List Price $75.00 Your Price $75.00
Cayman Vilanterol - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-20702-1
MFG.PART: 20702-1
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
Vilanterol is a long-acting agonist of the β2-adrenergic receptor (β2-AR). It selectively induces cAMP accumulation in CHO Cells expressing the β2-AR over the β1- and β3-ARs (EC50s = 0.4, 398, and 794 nM for the human receptors, respectively). Vilanterol inhibits contractions induced by electrical stimulation in isolated superfused guinea pig trachea strips. It inhibits bronchospasms induced by histamine (Item No. ) in guinea pigs when administered via nebulization (EC50 = 30 µM). Formulations containing vilanterol, in combination with fluticasone, have been used in the treatment of chronic obstructive pulmonary disease (COPD) and asthma.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
α1R-[[[6-[2-
CAS Number
503068-34-6
Synonyms
- GSK642444
- GW 642444
Molecular Formula
C24H33Cl2NO5
Formula Weight
486.4
Purity
≥98%
Formulation
A solution in ethanol
Solubility
- DMF: 30 mg/mL
- DMSO: 10 mg/mL
- Ethanol: 30 mg/mL
SMILES
ClC1=C(COCCOCCCCCCNC[C@H](O)C2=CC=C(O)C(CO)=C2)C(Cl)=CC=C1
InChi Code
InChI=1S/C24H33Cl2NO5/c25-21-6-5-7-22(26)20(21)17-32-13-12-31-11-4-2-1-3-10-27-15-24(30)18-8-9-23(29)19(14-18)16-28/h5-9,14,24,27-30H,1-4,10-13,15-17H2/t24-/m0/s1
InChi Key
DAFYYTQWSAWIGS-DEOSSOPVSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 2 years
| SKU | CAYM-20702-1 |
|---|---|
| Supplier Part Number | 20702-1 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | Y |
| CAS Number | 503068-34-6 |
| Energy Star | No |
| Green | No |
| Controlled | N |