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Cayman CPI-268456
List Price $36.00 Your Price $36.00
Cayman CPI-268456 - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-20973-1
MFG.PART: 20973-1
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
CPI-268456 is a ligand of bromodomain-containing protein 4 (BRD4). It binds to BRD4 (IC50 = <0.5 µM in a cell-free assay) and inhibits LPS-induced IL-6 secretion in THP-1 cells (IC50 = <0.5 µM).
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
(4S)-8-chloro-
CAS Number
1380087-86-4
Molecular Formula
C20H15Cl2N3O2
Formula Weight
400.3
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 30 mg/mL
- DMF:PBS (pH 7.2) (1:3): 0.25 mg/mL
- DMSO: 20 mg/mL
- Ethanol: 20 mg/mL
λmax
256 nm
SMILES
NC(C[C@@H]1N=C(C2=CC=C(Cl)C=C2)C3=C(C=CC(Cl)=C3)C4=C1ON=C4C)=O
InChi Code
InChI=1S/C20H15Cl2N3O2/c1-10-18-14-7-6-13(22)8-15(14)19(11-2-4-12(21)5-3-11)24-16(9-17(23)26)20(18)27-25-10/h2-8,16H,9H2,1H3,(H2,23,26)/t16-/m0/s1
InChi Key
RKYPLOAYXFDLOF-INIZCTEOSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Wet ice in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-20973-1 |
|---|---|
| Supplier Part Number | 20973-1 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 1380087-86-4 |
| Energy Star | No |
| Green | No |
| Controlled | N |