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Cayman SB-674042
List Price
$129.00
Your Price
$129.00
Cayman SB-674042 - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-21270-5
MFG.PART:
21270-5
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
SB-674042 is a potent and selective non-peptide orexin 1 receptor (OX1R) antagonist (Kd = 5.03 and 3.76 nM in whole cell binding and membrane-based assays, respectively).1 In calcium mobilization studies, it was >100-fold selective for OX1 over OX2 and did not show significant affinity for serotonergic, dopaminergic, adrenergic, or purinergic receptors at concentrations up to 10 µM.2
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
[5-(2-fluoro
CAS Number
483313-22-0
Molecular Formula
C24H21FN4O2S
Formula Weight
448.5
Purity
≥98%
Formulation(Request formulation change)
A crystalline solid
Solubility(Learn about Variance in Solubility)
- DMF: 30 mg/mL
- DMSO: 30 mg/mL
λmax
252 nm
SMILES
O=C(C1=C(C2=CC=CC=C2F)SC(C)=N1)N3[C@H](CC4=NN=C(C5=CC=CC=C5)O4)CCC3
InChi Code
InChI=1S/C24H21FN4O2S/c1-15-26-21(22(32-15)18-11-5-6-12-19(18)25)24(30)29-13-7-10-17(29)14-20-27-28-23(31-20)16-8-3-2-4-9-16/h2-6,8-9,11-12,17H,7,10,13-14H2,1H3/t17-/m0/s1
InChi Key
HYBZWVLPALMACV-KRWDZBQOSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-21270-5 |
|---|---|
| Supplier Part Number | 21270-5 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 483313-22-0 |
| Energy Star | No |
| Green | No |
| Controlled | N |