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Cayman L-Moses (hydrochloride)
List Price
$178.00
Your Price
$178.00
Cayman L-Moses (hydrochloride) - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-21288-5
MFG.PART:
21288-5
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
L-Moses is an inhibitor of the p300/CBP-associated factor (PCAF) bromodomain (Kd = 126 nM).1 It is selective for PCAF over GCN5 (Kd = 600 nM) and >4,500-fold selective for PCAF over BRD4. L-Moses displaces the PCAF bromodomain from histone H3.3 in a nanoBRET target engagement assay when used at a concentration of 5 μM.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
(1S,2S)-N1, N1-dimethyl- N2-(3-methyl- 1,2,4- triazolo [3,4-a] phthalazin- 6-yl)-1- phenyl-1,2- propane diamine, dihydro chloride
Synonyms
- L-45
Molecular Formula
C21H24N6 • 2HCl
Formula Weight
433.4
Purity
≥98%
Formulation(Request formulation change)
A crystalline solid
Solubility(Learn about Variance in Solubility)
- DMF: 25 mg/mL
- DMSO: 20 mg/mL
- Ethanol: 10 mg/mL
- PBS (pH 7.2): 10 mg/mL
λmax
233, 241, 557 nm
SMILES
CN(C)[C@@H](C1=CC=CC=C1)[C@H](C)NC(C2=CC=CC=C23)=NN4C3=NN=C4C.Cl.Cl
InChi Code
InChI=1S/C21H24N6.2ClH/c1-14(19(26(3)4)16-10-6-5-7-11-16)22-20-17-12-8-9-13-18(17)21-24-23-15(2)27(21)25-20;;/h5-14,19H,1-4H3,(H,22,25);2*1H/t14-,19+;;/m0../s1
InChi Key
PCQCTBXCEBIRAC-YRRRDGBXSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-21288-5 |
|---|---|
| Supplier Part Number | 21288-5 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 2922480-38-2 |
| Energy Star | No |
| Green | No |
| Controlled | N |