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Cayman SHA-68
List Price
$36.00
Your Price
$36.00
Cayman SHA-68 - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-21512-1
MFG.PART:
21512-1
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
SHA-68 is an antagonist of the neuropeptide S receptor (NPSR; IC50s = 22 and 23.8 nM for the NPSR Asn107 and NPSR Ile107 isoforms, respectively). It is selective for NPSR over a panel of 14 g protein-coupled receptors exhibiting no activity at a concentration of 10 μM. SHA-68 (50 mg/kg) reduces NPS-induced horizontal activity and vertical rearing and climbing in mice. SHA-68 also reduces conditioned reinstatement of cocaine seeking in rats.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
N-[(4-fluoro
CAS Number
847553-89-3
Molecular Formula
C26H24FN3O3
Formula Weight
445.5
Purity
≥95%
Formulation
A crystalline solid
Solubility
- DMF: 16 mg/mL
- DMSO: 14 mg/mL
- Ethanol: 20 mg/mL
- Ethanol:PBS (pH 7.2)(1:2): 0.33 mg/mL
SMILES
O=C(N1CC2N(C(OC2(C3=CC=CC=C3)C4=CC=CC=C4)=O)CC1)NCC5=CC=C(F)C=C5
InChi Code
InChI=1S/C26H24FN3O3/c27-22-13-11-19(12-14-22)17-28-24(31)29-15-16-30-23(18-29)26(33-25(30)32,20-7-3-1-4-8-20)21-9-5-2-6-10-21/h1-14,23H,15-18H2,(H,28,31)
InChi Key
SFRQIPRTNYHJHP-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-21512-1 |
|---|---|
| Supplier Part Number | 21512-1 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 847553-89-3 |
| Energy Star | No |
| Green | No |
| Controlled | N |