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Cayman Butabindide (oxalate)
List Price $918.00 Your Price $918.00
Cayman Butabindide (oxalate) - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-21610-50
MFG.PART: 21610-50
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
Butabindide is a potent inhibitor of cholecystokinin-inactivating peptidase/tripeptidyl peptidase 2 (CCK-inactivating peptidase/TPP-2; Ki = 7 nM).1 It is selective for CCK-inactivating peptidase/TPP-2 over a panel of serine proteases (Kis = >1 μM) as well as CCK receptors (Kis = >0.1 mm). Butabindide (0.1-100 μM) increases levels of CCK octapeptide (Item Nos. 24404 | 23371) in depolarized rat cerebral cortex slices. In vivo, butabindide inhibits CCK-inactivating peptidase/TPP-2 in mouse liver and brain (ID50s = 1.1 and 6.8 mg/kg, respectively). It also enhances CCK octapeptide-induced delay in gastric emptying and reduces food intake in mice.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
[S-(R*,R*)]-
CAS Number
185213-03-0
Molecular Formula
C17H25N3O2 • C2H2O4
Formula Weight
393.4
Purity
≥98%
Formulation(Request formulation change)
A crystalline solid
Solubility(Learn about Variance in Solubility)
- DMF: 1.6 mg/mL
- DMF:PBS (pH 7.2) (1:9): 0.1 mg/mL
λmax
250, 280, 288 nm
SMILES
O=C(NCCCC)[C@H]1N(C([C@@H](N)CC)=O)C2=CC=CC=C2C1.OC(C(O)=O)=O
InChi Code
InChI=1S/C17H25N3O2.C2H2O4/c1-3-5-10-19-16(21)15-11-12-8-6-7-9-14(12)20(15)17(22)13(18)4-2;3-1(4)2(5)6/h6-9,13,15H,3-5,10-11,18H2,1-2H3,(H,19,21);(H,3,4)(H,5,6)/t13-,15-;/m0./s1
InChi Key
KKMJFDVOXSGHBF-SLHAJLBXSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-21610-50 |
|---|---|
| Supplier Part Number | 21610-50 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 185213-03-0 |
| Energy Star | No |
| Green | No |
| Controlled | N |