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Cayman Salvinorin B Mesylate
List Price $107.00 Your Price $107.00
Cayman Salvinorin B Mesylate - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-22244-500
MFG.PART: 22244-500
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
Salvinorin B mesylate (Mesyl Sal B) is a selective κ-opioid receptor agonist that is more potent than salvinorin A (Item No. 11487) in CHO Cells transfected with the human κ-opioid receptor (EC50s = 30 and 40 nM, respectively).1,2 It is a mesylated version of salvinorin B (Item No. 11488) and is highly selective for κ-opioid receptors over µ- and δ-opioid receptors.1 In vitro, it increases dopamine uptake via the dopamine transporter (DAT) in an ERK1/2-dependent manner but does not alter expression of DAT on the cell membrane.3 In rats, it increases the pain threshold and blocks reinstatement of cocaine drug-seeking.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
(2S,4aR,6aR,
CAS Number
862073-79-8
Synonyms
- Divinorin B Mesylate
- Mesyl Sal B
- Sal B Mesylate
Molecular Formula
C22H28O9S
Formula Weight
468.5
Purity
≥95%
Formulation(Request formulation change)
A crystalline solid
Solubility(Learn about Variance in Solubility)
- DMF: 20 mg/mL
- DMSO: 20 mg/mL
- DMSO:PBS (pH 7.2) (1:7): 0.125 mg/mL
- Ethanol: slightly soluble
λmax
205 nm
SMILES
[H][C@@]12CC[C@@]([C@@]3([H])[C@@]1(C)C[C@@H](C4=COC=C4)OC2=O)(C)[C@H](C(OC)=O)C[C@H](OS(C)(=O)=O)C3=O
InChi Code
InChI=1S/C22H28O9S/c1-21-7-5-13-20(25)30-16(12-6-8-29-11-12)10-22(13,2)18(21)17(23)15(31-32(4,26)27)9-14(21)19(24)28-3/h6,8,11,13-16,18H,5,7,9-10H2,1-4H3/t13-,14-,15-,16-,18-,21-,22-/m0/s1
InChi Key
JPQCLBRBPPZECE-VOVNARLJSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Wet ice in continental US; may vary elsewhere
Stability
≥ 2 years
| SKU | CAYM-22244-500 |
|---|---|
| Supplier Part Number | 22244-500 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 862073-79-8 |
| Energy Star | No |
| Green | No |
| Controlled | N |