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Cayman ADL5859 (hydrochloride)
List Price
$228.00
Your Price
$228.00
Cayman ADL5859 (hydrochloride) - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-27796-10
MFG.PART:
27796-10
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
ADL5859 is a δ-opioid receptor agonist (Ki = 0.84 nM). It is selective for δ-opioid receptors over μ-opioid and κ-opioid receptors exhibiting 32 and 37% inhibition, respectively, in radioligand binding assays when used at a concentration of 10 μM. ADL5859 (3 mg/kg) completely reverses mechanical hyperalgesia induced by complete Freund’s adjuvant (CFA) in rats. It also decreases immobility time in the forced swim test in rats, indicating antidepressant-like activity.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
N,N-diethyl-4- (5-hydroxy spiro[2H-1- benzopyran- 2,4-piper idin]-4-yl)- benzamide, monohydro chloride
CAS Number
850173-95-4
Molecular Formula
C24H28N2O3 • HCl
Formula Weight
429.0
Purity
≥98%
Formulation
A solid
Solubility
- DMF: 3mg/mL
- DMSO: 10mg/mL
- DMSO:PBS (pH 7.2) (1:6): 0.14mg/mL
λmax
210, 252 nm
SMILES
O=C(N(CC)CC)C(C=C1)=CC=C1C2=CC3(CCNCC3)OC4=CC=CC(O)=C42.Cl
InChi Code
InChI=1S/C24H28N2O3.ClH/c1-3-26(4-2)23(28)18-10-8-17(9-11-18)19-16-24(12-14-25-15-13-24)29-21-7-5-6-20(27)22(19)21;/h5-11,16,25,27H,3-4,12-15H2,1-2H3;1H
InChi Key
ZFNLSWREIULTDO-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-27796-10 |
|---|---|
| Supplier Part Number | 27796-10 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | China |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 850173-95-4 |
| Energy Star | No |
| Green | No |
| Controlled | N |