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Cayman GLS1 Inhibitor
List Price $36.00 Your Price $36.00
Cayman GLS1 Inhibitor - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-28581-1
MFG.PART: 28581-1
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
GLS1 inhibitor is an inhibitor of glutaminase 1 (GLS1; IC50 = 0.021 μM). It inhibits the growth of NCI H1703 non-small cell lung cancer (NSCLC) cells in vitro (GI50 = 0.011 μM). GLS1 inhibitor (100 mg/kg) reduces tumor growth, increases tumor levels of glutamine, and decreases tumor levels of glutamate and aspartate in an NCI H1703 mouse xenograft model.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
αS-methoxy-N-
CAS Number
1832646-52-2
Molecular Formula
C19H21N7O2S
Formula Weight
411.5
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 20 mg/mL
- DMSO: 20 mg/mL
- DMSO:PBS (pH 7.2) (1:3): 0.25 mg/mL
λmax
252, 289 nm
SMILES
CO[C@H](C(NC1=NN=C(N[C@@H]2CCN(C3=CC=CN=N3)C2)S1)=O)C4=CC=CC=C4
InChi Code
InChI=1S/C19H21N7O2S/c1-28-16(13-6-3-2-4-7-13)17(27)22-19-25-24-18(29-19)21-14-9-11-26(12-14)15-8-5-10-20-23-15/h2-8,10,14,16H,9,11-12H2,1H3,(H,21,24)(H,22,25,27)/t14-,16+/m1/s1
InChi Key
KLQLQDLJJUAEGT-ZBFHGGJFSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Wet ice in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-28581-1 |
|---|---|
| Supplier Part Number | 28581-1 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 1832646-52-2 |
| Energy Star | No |
| Green | No |
| Controlled | N |