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Cayman DADLE
List Price
$36.00
Your Price
$36.00
Cayman DADLE - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-28928-1
MFG.PART:
28928-1
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
DADLE is a peptide agonist of δ-opioid receptors (Ki = 2.06 nM in a radioligand binding assay). It is selective for δ-opioid over κ-opioid receptors (Ki = 16,000 nM) but also agonizes μ-opioid receptors (Ki = 13.8 nM). DADLE inhibits electrically induced contractions in guinea pig myenteric plexus and mouse and rat vas deferens (IC50s = 8.9, 0.73, and 134 nM, respectively). It induces analgesia in the tail-flick and hot plate tests in mice (ED50s = 0.03 and 0.027 nmol per animal, i.c.v.).
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
L-tyrosyl-D-
CAS Number
63631-40-3
Synonyms
- [D-Ala2, D-Leu5]-Enkephalin
Molecular Formula
C29H39N5O7
Formula Weight
569.7
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 25 mg/mL
- DMSO: 25 mg/mL
- Ethanol: 3 mg/mL
- PBS (pH 7.2): 10 mg/mL
SMILES
OC1=CC=C(C[C@H](N)C(N[C@H](C)C(NCC(N[C@@H](CC2=CC=CC=C2)C(N[C@H](CC(C)C)C(O)=O)=O)=O)=O)=O)C=C1
InChi Code
InChI=1S/C29H39N5O7/c1-17(2)13-24(29(40)41)34-28(39)23(15-19-7-5-4-6-8-19)33-25(36)16-31-26(37)18(3)32-27(38)22(30)14-20-9-11-21(35)12-10-20/h4-12,17-18,22-24,35H,13-16,30H2,1-3H3,(H,31,37)(H,32,38)(H,33,36)(H,34,39)(H,40,41)/t18-,22+,23+,24-/m1/s1
InChi Key
ZHUJMSMQIPIPTF-IBURTVSXSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-28928-1 |
|---|---|
| Supplier Part Number | 28928-1 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | China |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 63631-40-3 |
| Energy Star | No |
| Green | No |
| Controlled | N |