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Cayman DY 268
List Price $128.00 Your Price $128.00
Cayman DY 268 - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-29475-5
MFG.PART: 29475-5
UNSPSC: 12352200
Manufacturer: Cayman


Product Description
DY 268 is a farnesoid X receptor (FXR) antagonist (IC50 = 7.5 nM in a time-resolved FRET assay).1 It inhibits FXR transactivation in a cell-based assay with an IC50 value of 468 nM.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
1-[(3-methoxy phenyl) methyl]-N-[4- methyl-3-(4- morpholinyl sulfonyl) phenyl]-3-(4- methylphenyl)- 1H-pyrazole- 4-carboxamide
CAS Number
1609564-75-1
Molecular Formula
C30H32N4O5S
Formula Weight
560.7
Purity
≥98%
Formulation(Request formulation change)
A solid
Solubility(Learn about Variance in Solubility)
- DMSO: soluble
λmax
250 nm
SMILES
CC(C=C1)=CC=C1C2=NN(CC3=CC=CC(OC)=C3)C=C2C(NC4=CC=C(C)C(S(N5CCOCC5)(=O)=O)=C4)=O
InChi Code
InChI=1S/C30H32N4O5S/c1-21-7-10-24(11-8-21)29-27(20-33(32-29)19-23-5-4-6-26(17-23)38-3)30(35)31-25-12-9-22(2)28(18-25)40(36,37)34-13-15-39-16-14-34/h4-12,17-18,20H,13-16,19H2,1-3H3,(H,31,35)
InChi Key
KQSPAAPFKIEUGH-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-29475-5 |
|---|---|
| Supplier Part Number | 29475-5 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 1609564-75-1 |
| Energy Star | No |
| Green | No |
| Controlled | N |

