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Cayman VCP171
List Price $502.00 Your Price $502.00
Cayman VCP171 - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-30309-25
MFG.PART: 30309-25
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
VCP171 is a positive allosteric modulator of adenosine A1 receptors (EC50 = 15.8 μM in a kinetic assay measuring agonist dissociation).1. It reduces AMPA receptor-mediated evoked excitatory postsynaptic currents (eEPSCs) in lamina I and lamina II neurons in a rat model of neuropathic pain (EC50s = 1.995 and 0.251 μM, respectively) to a greater extent than in sham control animals (EC50s = 2.512 and 0.631 μM, respectively).2
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
[2-amino-4-
CAS Number
1018830-99-3
Molecular Formula
C18H12F3NOS
Formula Weight
347.4
Purity
≥98%
Formulation(Request formulation change)
A crystalline solid
Solubility(Learn about Variance in Solubility)
- DMF: 30 mg/mL
- DMSO: 30 mg/mL
- DMSO:PBS (pH 7.2) (1:6): 0.14 mg/mL
- Ethanol: 10 mg/mL
λmax
210, 241 nm
SMILES
NC1=C(C(C2=CC=CC=C2)=O)C(C3=CC(C(F)(F)F)=CC=C3)=CS1
InChi Code
InChI=1S/C18H12F3NOS/c19-18(20,21)13-8-4-7-12(9-13)14-10-24-17(22)15(14)16(23)11-5-2-1-3-6-11/h1-10H,22H2
InChi Key
HNHLVOBHWXLIGP-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Wet ice in continental US; may vary elsewhere
Stability
≥ 2 years
| SKU | CAYM-30309-25 |
|---|---|
| Supplier Part Number | 30309-25 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 1018830-99-3 |
| Energy Star | No |
| Green | No |
| Controlled | N |