We use cookies to make your experience better. To comply with the new e-Privacy directive, we need to ask for your consent to set the cookies. Learn more.
Cayman (+)-JQ1 PA
List Price
$153.00
Your Price
$153.00
Cayman (+)-JQ1 PA - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-30414-5
MFG.PART:
30414-5
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
(+)-JQ1 PA is a clickable form of the bromodomain and extraterminal domain (BET) inhibitor (+)-JQ1 (Item Nos. 11187 | 9002910).1 (+)-JQ1 PA binds to bromodomain-containing protein 4 (BRD4) and displaces it from Myc in a ChIP-qPCR assay. It reduces proliferation of MV4-11 cells (IC50 = 10.4 nM).
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
(6S)-4-(4-
CAS Number
2115701-93-2
Synonyms
- Click Tag™ (+)-JQ1 PA
Molecular Formula
C22H20ClN5OS
Formula Weight
437.9
Purity
≥98%
Formulation(Request formulation change)
A crystalline solid
Solubility(Learn about Variance in Solubility)
- DMF: 30 mg/mL
- DMSO: 30 mg/mL
- DMSO:PBS (pH 7.2) (1:6): 0.14 mg/mL
- Ethanol: 25 mg/mL
λmax
255 nm
SMILES
CC1=C(C)C(C(C2=CC=C(Cl)C=C2)=N[C@@H](CC(NCC#C)=O)C3=NN=C(C)N34)=C4S1
InChi Code
InChI=1S/C22H20ClN5OS/c1-5-10-24-18(29)11-17-21-27-26-14(4)28(21)22-19(12(2)13(3)30-22)20(25-17)15-6-8-16(23)9-7-15/h1,6-9,17H,10-11H2,2-4H3,(H,24,29)/t17-/m0/s1
InChi Key
ZLSCJWMPQYKVKU-KRWDZBQOSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-30414-5 |
|---|---|
| Supplier Part Number | 30414-5 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | China |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 2115701-93-2 |
| Energy Star | No |
| Green | No |
| Controlled | N |