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Cayman Remoxipride (hydrochloride)
List Price
$41.00
Your Price
$41.00
Cayman Remoxipride (hydrochloride) - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-30971-1
MFG.PART:
30971-1
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
Remoxipride is an atypical antipsychotic and dopamine D2 receptor antagonist (Ki = 0.2 µM). It is selective for the dopamine D2 receptor over a panel of 33 receptors, neurotransmitter transporters, and ion channels at 10 µM but does inhibit the sigma (σ) receptor (Ki = 0.065 µM). Remoxipride (2-20 µmol/kg, i.p.) increases striatal 3,4-dihydroxyphenylacetic acid (DOPAC) and homovanillic acid (HVA) levels in rats. It inhibits apomorphine-induced stereotypy and hyperactivity in rats with ED50 values of 5.6 and 0.8 µmol/kg, respectively. Formulations containing remoxipride have previously been used in the treatment of schizophrenia.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
3-bromo-N-
CAS Number
73220-03-8
Molecular Formula
C16H23BrN2O3 • HCl
Formula Weight
407.7
Purity
≥98%
Formulation
A crystalline solid
Solubility
- Water: 100 mm
SMILES
BrC1=CC=C(OC)C(C(NC[C@H]2N(CC)CCC2)=O)=C1OC.Cl
InChi Code
InChI=1S/C16H23BrN2O3.ClH/c1-4-19-9-5-6-11(19)10-18-16(20)14-13(21-2)8-7-12(17)15(14)22-3;/h7-8,11H,4-6,9-10H2,1-3H3,(H,18,20);1H/t11-;/m0./s1
InChi Key
WCPXLMIPGMFZMY-MERQFXBCSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-30971-1 |
|---|---|
| Supplier Part Number | 30971-1 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 73220-03-8 |
| Energy Star | No |
| Green | No |
| Controlled | N |