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Cayman Mesoridazine
List Price $90.00 Your Price $90.00
Cayman Mesoridazine - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-31370-25
MFG.PART: 31370-25
UNSPSC: 12352200
Manufacturer: Cayman


Product Description
Mesoridazine is an active metabolite of the typical antipsychotic thioridazine (Item No. 14400).1,2 It is formed via sulfoxidation of thioridazine by the cytochrome P450 (CYP) isoform CYP2D6 in human liver microsomes.3 It binds to histamine H1, dopamine D2, muscarinic acetylcholine, and α1- and α2-adrenergic receptors (Kds = 1.8, 19, 69, 2, and 1,600 nM, respectively).2 Mesoridazine (10, 30, and 45 mg/kg, i.p.) prevents mescaline-induced hyperactivity in mice.4
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
10-[2-(1- methyl-2- piperidinyl) ethyl]-2- (methyl sulfinyl)- 10H-pheno thiazine
CAS Number
5588-33-0
Synonyms
- NSC 186066
Molecular Formula
C21H26N2OS2
Formula Weight
386.6
Purity
≥95%
Formulation(Request formulation change)
A solution in acetonitrile
Solubility(Learn about Variance in Solubility)
- Acetonitrile: slightly soluble
- DMSO: slightly, heated
- Methanol: slightly soluble
SMILES
O=S(C)C1=CC=C2SC3=C(N(CCC4N(CCCC4)C)C2=C1)C=CC=C3O=S(C)C1=CC=C2SC3=C(N(CCC4N(CCCC4)C)C2=C1)C=CC=C3
InChi Code
InChI=1S/C21H26N2OS2/c1-22-13-6-5-7-16(22)12-14-23-18-8-3-4-9-20(18)25-21-11-10-17(26(2)24)15-19(21)23/h3-4,8-11,15-16H,5-7,12-14H2,1-2H3
InChi Key
SLVMESMUVMCQIY-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 2 years
| SKU | CAYM-31370-25 |
|---|---|
| Supplier Part Number | 31370-25 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | Canada |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | Y |
| CAS Number | 5588-33-0 |
| Energy Star | No |
| Green | No |
| Controlled | N |

