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Cayman (S)-WAY-100135 (hydrochloride)
List Price $134.00 Your Price $134.00
Cayman (S)-WAY-100135 (hydrochloride) - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-32851-10
MFG.PART: 32851-10
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
(S)-WAY-100135 is an antagonist of the serotonin (5-HT) receptor subtype 5-HT1A (IC50 = 15.5 nM in a radioligand binding assay using rat hippocampus). It is selective for 5-HT1A over 5-HT1B, 5-HT1C, and 5-HT2 receptors, as well as dopamine D1 and D2, and α1-, α2-, and β-adrenergic receptors (IC50s = >1 µM for all). (S)-WAY-100135 (10 mg/kg) increases the number of entries into and percentage of time spent in the open arms of the elevated plus maze in mice, indicating anxiolytic-like activity.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
(αS)-N-(1,1-dimethylethyl)-4-(2-methoxyphenyl)-α-phenyl-1-piperazinepropanamide, dihydrochloride
CAS Number
149007-54-5
Molecular Formula
C24H33N3O2 • 2HCl
Formula Weight
468.5
Purity
≥98%
Formulation
A solid
Solubility
- DMSO: 100 mm
- Water: 10 mm
SMILES
COC1=C(N2CCN(CC2)C[C@H](C3=CC=CC=C3)C(NC(C)(C)C)=O)C=CC=C1.Cl.Cl
InChi Code
InChI=1S/C24H33N3O2.2ClH/c1-24(2,3)25-23(28)20(19-10-6-5-7-11-19)18-26-14-16-27(17-15-26)21-12-8-9-13-22(21)29-4;;/h5-13,20H,14-18H2,1-4H3,(H,25,28);2*1H/t20-;;/m1../s1
InChi Key
VJGZNBYDSDEOED-FAVHNTAZSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-32851-10 |
|---|---|
| Supplier Part Number | 32851-10 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | Y |
| CAS Number | 149007-54-5 |
| Energy Star | No |
| Green | No |
| Controlled | N |