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Cayman Deslorelin (acetate)
List Price
$448.00
Your Price
$448.00
Cayman Deslorelin (acetate) - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-34041-25
MFG.PART:
34041-25
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
Deslorelin is a peptide agonist of gonadotropin-releasing hormone (GnRH).1 It binds to the GnRH receptor (GnRHR) with a Ki value of 0.1 nM. Deslorelin decreases testicular volume, semen volume, sperm motility, and total sperm count, as well as increases the percentage of abnormal sperm, in dogs when administered via a subcutaneous implant at doses of 3, 6, and 12 mg/kg.2 It decreases disease severity and plasma levels of estradiol, 17-hydroxyprogesterone, and androstenedione in ferrets with adrenocortical disease (ACD) when administered at doses ranging from 3 to 4.41 mg/kg per implant.3 Deslorelin (4.7 mg/implant per animal) suppresses ovulation and estrus in cats.4 Formulations containing deslorelin have been used in the management of ACD in ferrets and ovulation regulation and artificial insemination in horses.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
6-D-tryptophan-
CAS Number
1642579-30-3
Synonyms
- D-Trp6-Pro9-des-Gly10-GnRH ethylamide
- pGlu-His-Trp-Ser-Tyr-D-Trp-Leu-Arg-Pro-NHEt
Molecular Formula
C64H83N17O12 • XC2H4O2
Formula Weight
1282.5
Purity
≥98%
Formulation(Request formulation change)
A solid
Solubility(Learn about Variance in Solubility)
- DMF: 5 mg/mL
- DMSO: 5 mg/mL
- Ethanol: 10 mg/mL
λmax
219 nm
SMILES
OC(C=C1)=CC=C1C[C@H](NC([C@H](CO)NC([C@@H](NC([C@@H](NC([C@H]2NC(CC2)=O)=O)CC3=CN=CN3)=O)CC4=CNC5=CC=CC=C45)=O)=O)C(N[C@@H](C(N[C@@H](CC(C)C)C(N[C@@H](CCCNC(N)=N)C(N6[C@@H](CCC6)C(NCC)=O)=O)=O)=O)CC7=CNC8=CC=CC=C78)=O.CC(O)=O
InChi Code
InChI=1S/C64H83N17O12.C2H4O2/c1-4-68-62(92)53-16-10-24-81(53)63(93)46(15-9-23-69-64(65)66)74-56(86)47(25-35(2)3)75-58(88)49(27-37-30-70-43-13-7-5-11-41(37)43)77-57(87)48(26-36-17-19-40(83)20-18-36)76-61(91)52(33-82)80-59(89)50(28-38-31-71-44-14-8-6-12-42(38)44)78-60(90)51(29-39-32-67-34-72-39)79-55(85)45-21-22-54(84)73-45;1-2(3)4/h5-8,11-14,17-20,30-32,34-35,45-53,70-71,82-83H,4,9-10,15-16,21-29,33H2,1-3H3,(H,67,72)(H,68,92)(H,73,84)(H,74,86)(H,75,88)(H,76,91)(H,77,87)(H,78,90)(H,79,85)(H,80,89)(H4,65,66,69);1H3,(H,3,4)/t45-,46-,47-,48-,49+,50-,51-,52-,53-;/m0./s1
InChi Key
LYCYLGFSIXIXAB-NUZRHMIVSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-34041-25 |
|---|---|
| Supplier Part Number | 34041-25 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | China |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 1642579-30-3 |
| Energy Star | No |
| Green | No |
| Controlled | N |