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Cayman Dabigatran etexilate (mesylate)
List Price $513.00 Your Price $513.00
Cayman Dabigatran etexilate (mesylate) - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-35248-1
MFG.PART: 35248-1
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
Dabigatran etexilate is a prodrug form of the thrombin inhibitor dabigatran (Item No. 17133).1 It inhibits thrombin-induced platelet aggregation in isolated rabbit platelets (IC50 = 0.337 µM) and inhibits thrombus formation in a rat model of venous thrombosis (ED50 = 7.8 µmol/kg). Formulations containing dabigatran etexilate have been used to reduce the risk of stroke and systemic embolism in patients with non-valvular atrial fibrillation and in the treatment and prevention of deep vein thrombosis (DVT) and pulmonary embolism.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
N-[[2-[[[4-
CAS Number
872728-81-9
Synonyms
- BIBR 1048MS
Molecular Formula
C34H41N7O5 • CH3SO3H
Formula Weight
723.8
Purity
≥98%
Formulation(Request formulation change)
A solid
Solubility(Learn about Variance in Solubility)
- DMF: 10 mg/mL
- DMSO: 10 mg/mL
- Ethanol: 5 mg/mL
- PBS (pH 7.2): 0.3 mg/mL
λmax
226, 344 nm
SMILES
O=C(NC(C1=CC=C(NCC2=NC3=CC(C(N(CCC(OCC)=O)C4=CC=CC=N4)=O)=CC=C3N2C)C=C1)=N)OCCCCCC.O=S(O)(C)=O
InChi Code
InChI=1S/C34H41N7O5.CH4O3S/c1-4-6-7-10-21-46-34(44)39-32(35)24-12-15-26(16-13-24)37-23-30-38-27-22-25(14-17-28(27)40(30)3)33(43)41(20-18-31(42)45-5-2)29-11-8-9-19-36-29;1-5(2,3)4/h8-9,11-17,19,22,37H,4-7,10,18,20-21,23H2,1-3H3,(H2,35,39,44);1H3,(H,2,3,4)
InChi Key
XETBXHPXHHOLOE-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-35248-1 |
|---|---|
| Supplier Part Number | 35248-1 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | China |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 872728-81-9 |
| Energy Star | No |
| Green | No |
| Controlled | N |