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Cayman Met-Enkephalinamide (trifluoroacetate salt)
List Price $329.00 Your Price $329.00
Cayman Met-Enkephalinamide (trifluoroacetate salt) - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-36081-50
MFG.PART: 36081-50
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
Met-Enkephalinamide is a peptide opioid receptor agonist and derivative of Met-enkephalin (Item No. 23284).1,2 It binds to opioid receptors in rat cerebellum homogenates (IC50 = 0.2 µM) and reduces the twitch height in electrically stimulated isolated guinea pig ileum and isolated mouse vas deferens. Met-Enkephalinamide (300 µg/animal) induces analgesia in the hot plate and tail-flick tests in rats, effects that can be reversed by administration of the opioid receptor antagonist naloxone.3
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
L-tyrosyl
Synonyms
- [Met5]-Enkephalin amide
- Methionine-Enkephalin amide
- H-Tyr-Gly-Gly-Phe-Met-NH2
- H-YGGFM-NH2
Molecular Formula
C27H36N6O6S • XCF3COOH
Formula Weight
572.7
Purity
≥98%
Formulation(Request formulation change)
A solid
Solubility(Learn about Variance in Solubility)
- DMF: 2 mg/mL
- DMSO: 10 mg/mL
- Ethanol: 3 mg/mL
- PBS (pH 7.2): 2 mg/mL
SMILES
O=C(N[C@H](C(N)=O)CCSC)[C@@H](NC(CNC(CNC([C@@H](N)CC(C=C1)=CC=C1O)=O)=O)=O)CC2=CC=CC=C2.OC(C(F)(F)F)=O
InChi Code
InChI=1S/C27H36N6O6S.C2HF3O2/c1-40-12-11-21(25(29)37)33-27(39)22(14-17-5-3-2-4-6-17)32-24(36)16-30-23(35)15-31-26(38)20(28)13-18-7-9-19(34)10-8-18;3-2(4,5)1(6)7/h2-10,20-22,34H,11-16,28H2,1H3,(H2,29,37)(H,30,35)(H,31,38)(H,32,36)(H,33,39);(H,6,7)/t20-,21-,22-;/m0./s1
InChi Key
RZLKVUJHGWGFHT-SGIIKHNDSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-36081-50 |
|---|---|
| Supplier Part Number | 36081-50 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | China |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| Energy Star | No |
| Green | No |
| Controlled | N |