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Cayman A2764 (hydrochloride)
List Price $227.00 Your Price $227.00
Cayman A2764 (hydrochloride) - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-36943-100
MFG.PART: 36943-100
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
A2764 is an inhibitor of the two-pore domain potassium channel K2P18.1/TRESK (IC50 = 11.8 µM in ionomycin-stimulated Xenopus oocytes expressing the mouse receptor).1 It is selective for K2P18.1/TRESK over K2P2.1/TREK1, K2P10.1/TREK2, K2P4.1/TRAAK, K2P3.1/TASK1, K2P3.2/TASK2, K2P3.3/TASK3, K2P16.1/TALK1, and K2P13.1/THIK1 at 100 µM. A2764 (100 µM) inhibits basal potassium currents in isolated mouse dorsal root ganglion neurons.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
2-[(5-chloro-
CAS Number
861038-72-4
Molecular Formula
C15H19ClN2O • 2HCl
Formula Weight
351.7
Purity
≥98%
Formulation(Request formulation change)
A solid
Solubility(Learn about Variance in Solubility)
- DMSO: Slightly soluble
- Ethanol: Slightly soluble
- PBS (pH 7.2): 5 mg/mL
λmax
244 nm
SMILES
CCN(CC)CCOC1=CC=C(Cl)C2=C1N=CC=C2.Cl.Cl
InChi Code
InChI=1S/C15H19ClN2O.2ClH/c1-3-18(4-2)10-11-19-14-8-7-13(16)12-6-5-9-17-15(12)14;;/h5-9H,3-4,10-11H2,1-2H3;2*1H
InChi Key
ZVRDPULCSHGKBD-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-36943-100 |
|---|---|
| Supplier Part Number | 36943-100 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | China |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 861038-72-4 |
| Energy Star | No |
| Green | No |
| Controlled | N |