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Cayman AM0902
List Price $163.00 Your Price $163.00
Cayman AM0902 - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-37290-10
MFG.PART: 37290-10
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
AM0902 is a transient receptor potential ankyrin 1 (TRPA1) antagonist (IC50 = 0.131 µM for the human receptor in a calcium mobilization assay).1 It is selective for human TRPA1 over human transient receptor potential vanilloid 1 (TRPV1) and TRPV4, rat TRPV1, TRPV3, and transient receptor potential melastatin 8 (TRPM8), and a panel of 40 additional targets at 10 µM. In vivo, AM0902 (10 and 30 mg/kg) reduces the number of tail flinches induced by the TRPA1 agonist allyl isothiocyanate (AITC) in rats.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
1-[[3-[2-(4-
CAS Number
1883711-97-4
Molecular Formula
C17H15ClN6O2
Formula Weight
370.8
Purity
≥98%
Formulation(Request formulation change)
A solid
Solubility(Learn about Variance in Solubility)
- DMSO: Soluble
λmax
214 nm
SMILES
O=C1C2=C(N=CN2C)N=CN1CC3=NC(CCC4=CC=C(Cl)C=C4)=NO3
InChi Code
InChI=1S/C17H15ClN6O2/c1-23-9-19-16-15(23)17(25)24(10-20-16)8-14-21-13(22-26-14)7-4-11-2-5-12(18)6-3-11/h2-3,5-6,9-10H,4,7-8H2,1H3
InChi Key
AWJBWNUUODWOKQ-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-37290-10 |
|---|---|
| Supplier Part Number | 37290-10 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 1883711-97-4 |
| Energy Star | No |
| Green | No |
| Controlled | N |