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Cayman Rpn-13 Inhibitor TCL1, 1 mg
List Price
$32.00
Your Price
$32.00
Cayman Rpn-13 Inhibitor TCL1, 1 mg-CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-43982-1
MFG.PART:
43982-1
UNSPSC:
41106300
Manufacturer:
Cayman
Product Description
Rpn-13 inhibitor TCL1 is an inhibitor of UDP-galactopyranose mutase (UGM), also known as RfbD (Ki = 1.1 µM for the K. pneumoniae enzyme).1 It also binds to proteasomal ubiquitin receptor ADRM1, also known as proteasome regulatory particle non-ATPase 13 (Rpn-13; Kd = ~26 µM).2 Rpn-13 inhibitor TCL1 decreases growth of M. tuberculosis and M. smegmatis in a disk diffusion assay (MICs = 9.3 and 9.4 µg/mL, respectively).1
WARNING This product is not for human or veterinary use.
Technical Information
| Formal Name | 3-[(4bromophenyl)methyl]-6-(4-chlorophenyl)-7H-1,2,4-triazolo[3,4-b][1,3,4]thiadiazine-7-acetic acid |
| CAS Number | 875165-39-2 |
| Synonyms |
|
| Molecular Formula | C19H14BrClN4O2S |
| Formula Weight | 477.8 |
| Purity | ≥98% |
| Formulation(Request formulation change) | A solid |
| Solubility(Learn about Variance in Solubility) | DMSO: Slightly soluble: 0.1-1 mg/mL |
| SMILES | BrC1=CC=C(CC2=NN=C(SC3CC(O)=O)N2N=C3C4=CC=C(C=C4)Cl)C=C1 |
| InChi Code | InChI=1S/C19H14BrClN4O2S/c20-13-5-1-11(2-6-13)9-16-22-23-19-25(16)24-18(15(28-19)10-17(26)27)12-3-7-14(21)8-4-12/h1-8,15H,9-10H2,(H,26,27) |
| InChi Key | BWGPJTANFXCCTH-UHFFFAOYSA-N |
Shipping & Storage Information
| Storage | -20°C |
| Shipping | Room temperature in continental US; may vary elsewhere |
| Stability | ≥ 4 years |
| SKU | CAYM-43982-1 |
|---|---|
| Supplier Part Number | 43982-1 |
| UM | EA |
| UNSPSC | 41106300 |
| Manufacturer | Cayman |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 875165-39-2 |
| Energy Star | No |
| Green | No |
| Controlled | N |