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Cayman Landiolol (hydrochloride), 10 mg
List Price
$53.00
Your Price
$53.00
Cayman Landiolol (hydrochloride), 10 mg-CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-44229-10
MFG.PART:
44229-10
UNSPSC:
12352211
Manufacturer:
Cayman
Product Description
Landiolol is an antagonist of the β1-adrenergic receptor (β1-AR).1 It selectively induces relaxation of isolated and perfused guinea pig atrial strips that endogenously express β1-ARs over isolated and perfused guinea pig tracheal strips that endogenously express β2-ARs (PA2s = 6.59 and 4.18, respectively). Infusion of landiolol (10 µg/kg per minute) inhibits tachycardia induced by isoproterenol (Item No. 15592) in dogs. Formulations containing landiolol have been used in the treatment of supraventricular tachycardia.
WARNING This product is not for human or veterinary use.
Technical Information
| Formal Name | 4-[(2S)-2- |
| CAS Number | 144481-98-1 |
| Synonyms |
|
| Molecular Formula | C25H39N3O8 • HCl |
| Formula Weight | 546.1 |
| Purity | ≥98% |
| Formulation(Request formulation change) | A solid |
| Solubility(Learn about Variance in Solubility) | DMSO: Sparingly soluble: 1-10 mg/mLEthanol: Slightly soluble: 0.1-1 mg/mLPBS (pH 7.2): Sparingly soluble: 1-10 mg/mL |
| SMILES | CC(C)(OC1)O[C@@H]1COC(CCC2=CC=C(C=C2)OC[C@@H](O)CNCCNC(N3CCOCC3)=O)=O.Cl |
| InChi Code | InChI=1S/C25H39N3O8.ClH/c1-25(2)35-18-22(36-25)17-34-23(30)8-5-19-3-6-21(7-4-19)33-16-20(29)15-26-9-10-27-24(31)28-11-13-32-14-12-28;/h3-4,6-7,20,22,26,29H,5,8-18H2,1-2H3,(H,27,31);1H/t20-,22+;/m0./s1 |
| InChi Key | DLPGJHSONYLBKP-IKGOIYPNSA-N |
Shipping & Storage Information
| Storage | -20°C |
| Shipping | Room temperature in continental US; may vary elsewhere |
| Stability | ≥ 4 years |
| SKU | CAYM-44229-10 |
|---|---|
| Supplier Part Number | 44229-10 |
| UM | EA |
| UNSPSC | 12352211 |
| Manufacturer | Cayman |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | China |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 144481-98-1 |
| Energy Star | No |
| Green | No |
| Controlled | N |