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Cayman TUG-469, 10 mg
List Price $28.00 Your Price $28.00
Cayman TUG-469, 10 mg-CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-44272-10
MFG.PART: 44272-10
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
TUG-469 is an agonist of free fatty aid receptor 1 (FFAR1/GPR40).1 It induces calcium mobilization in a reporter assay using cells expressing human FFAR1/GPR40 (EC50 = 18.6 nM). TUG-469 (10 µM) induces insulin secretion in INS-1E insulinoma cells. It inhibits increases in blood glucose levels in a glucose tolerance test (GTT) in mice when administered at a dose of 5 mg/kg.2
WARNING This product is not for human or veterinary use.
Technical Information
| Formal Name | 4-[[(2′-methyl[1,1′-biphenyl]-3-yl)methyl]amino]-benzenepropanoic acid |
| CAS Number | 1236109-67-3 |
| Molecular Formula | C23H23NO2 |
| Formula Weight | 345.4 |
| Purity | ≥98% |
| Formulation(Request formulation change) | A solid |
| Solubility(Learn about Variance in Solubility) | DMSO: Sparingly soluble: 1-10 mg/mLEthanol: Slightly soluble: 0.1-1 mg/mL |
| SMILES | O=C(CCC1=CC=C(NCC2=CC(C3=C(C)C=CC=C3)=CC=C2)C=C1)O |
| InChi Code | InChI=1S/C23H23NO2/c1-17-5-2-3-8-22(17)20-7-4-6-19(15-20)16-24-21-12-9-18(10-13-21)11-14-23(25)26/h2-10,12-13,15,24H,11,14,16H2,1H3,(H,25,26) |
| InChi Key | RUPXKSLKGSSZCP-UHFFFAOYSA-N |
Shipping & Storage Information
| Storage | -20°C |
| Shipping | Room temperature in continental US; may vary elsewhere |
| Stability | ≥ 4 years |
| SKU | CAYM-44272-10 |
|---|---|
| Supplier Part Number | 44272-10 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | China |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 1236109-67-3 |
| Energy Star | No |
| Green | No |
| Controlled | N |