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Cayman Tianeptine Metabolite MC5
List Price $186.00 Your Price $186.00
Cayman Tianeptine Metabolite MC5 - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART: CAYM-36694-1
MFG.PART: 36694-1
UNSPSC: 12352200
Manufacturer: Cayman
Product Description
Tianeptine metabolite MC5 is an active metabolite of the atypical antidepressant tianeptine (Item No. 17561).1 It is formed from tianeptine by β-oxidation.2 Tianeptine metabolite MC5 selectively induces g protein activation in bioluminescence resonance energy transfer (BRET) assays using HEK293T cells expressing the human μ-opioid receptor (MOR) over the human δ-opioid receptor (DOR; EC50s = 0.454 and >100 µM, respectively).1 It decreases immobility in the forced swim test in wild-type mice, but not MOR knockout mice, indicating MOR-dependent antidepressant-like activity when administered at a dose of 30 mg/kg.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
5-[(3-chloro-
CAS Number
115220-11-6
Molecular Formula
C19H20ClN2O4S • Na
Formula Weight
430.9
Purity
≥98%
Formulation(Request formulation change)
A solid
Solubility(Learn about Variance in Solubility)
- Dichloromethane: Slightly soluble
- DMSO: Slightly soluble
- Methanol: Slightly soluble
SMILES
O=C(CCCCNC1C2=C(N(S(=O)(C3=CC(Cl)=CC=C31)=O)C)C=CC=C2)[O-].[Na+]
InChi Code
InChI=1S/C19H21ClN2O4S.Na/c1-22-16-7-3-2-6-14(16)19(21-11-5-4-8-18(23)24)15-10-9-13(20)12-17(15)27(22,25)26;/h2-3,6-7,9-10,12,19,21H,4-5,8,11H2,1H3,(H,23,24);/q;+1/p-1
InChi Key
GBYSEZGRQUELJJ-UHFFFAOYSA-M
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-36694-1 |
|---|---|
| Supplier Part Number | 36694-1 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Y |
| CountryOfOrigin | China |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 5 |
| Hazardous | N |
| CAS Number | 104732-22-1 |
| Energy Star | No |
| Green | No |
| Controlled | N |